http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CS-203083-B2
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_f07293d4b34d8372fb0775181fef9d23 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D495-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D495-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D333-36 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-55 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-551 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D495-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D495-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D333-36 |
| filingDate | 1975-02-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8fe55b7b362e3fa8f2c11e701d6d8fca http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f66c4333b93ccce26db84aaa2fbc1a38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fdbc00857b2425017d3d5d9407a74fd1 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_15d939ccea8e5fb41ed4485c8295c8af |
| publicationDate | 1981-02-27-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | CS-203083-B2 |
| titleOfInvention | Method of producing novel substituted 6-aryl-4h-o-triazolo/3,4-c/thieno/2,3-e/1,4-diazepines |
| abstract | 1497527 Heterocyclic-fused 1,4-diazepine derivatives BOEHRINGER INGELHEIM GmbH 3 March 1975 [20 July 1974 24 Sept 1974 21 Dec 1974] 27236/77 Divided out of 1490269 Heading C2C The invention comprises compounds of Formula (I) wherein R 1 is H, Cl, Br or C 1-4 alkyl; R 2 is H, F, Cl, Br, NO 2 or CF 3 ; R 3 is Cl, Br, C 1-3 alkoxy or alkylthio, C 3-6 cycloalkyl or cycloalkenyl, or a 5- or 6-membered heterocyclic ring; and (except where R 3 is an S-containing ring) their acid addition salts. In examples, (I) are prepared by (a) heating the hydrazides (VII) (b) reacting the unacylated analogue of (VII) with R 1 -COCl, (c) reacting the 2-SH*, -SMe or -OEt (de-acylhydrazide) analogues of (VII) with R 1 CONHNH 2 , or (d) converting one substitutent (R 3 ) into another; (VII) are prepared by reacting the 2-SH compounds* with R 1 CONHNH 2 . Therapeutic compositions having anxiolytic, tensiolytic, muscle-relaxing and anticonvulsive activity, and which increase the intake of food in warm-blooded animals, comprise compounds of the above Formula (I). They may be administered orally, parenterally or rectally, and may contain other active compounds such as spasmolytics or beta-receptor blockers. |
| priorityDate | 1974-03-02-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 73.