http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CO-5690582-A2
Outgoing Links
Predicate | Object |
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assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_a693232b92910547c898db10feb83fef |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-426 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D277-46 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-24 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-28 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-426 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D277-46 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-28 |
filingDate | 2006-04-25-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ac66dcd14713780c279d2e08cc4b56d5 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_de75c9a4c0686994115357c204edda76 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_59c97224381e363224e2b333075fc5fd |
publicationDate | 2006-10-31-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | CO-5690582-A2 |
titleOfInvention | DERIVATIVES OF N-TIAZOL-2-IL-BENZAMIDA |
abstract | 1.- Use of a compound of formula I: wherein R1 and R6 are, independently, hydrogen, C1-6 alkyl or halogen; R2-R5 are independently selected from the group consisting of: hydrogen, halogen, cyano, OH, NH2, nitro, C1-6 alkyl, aryl, arylC1-6 alkyl, heteroarylC1-6 alkyl, C3-8 cycloalkyl, C3-8 cycloalkyl-C1-6 alkyl, C1-6 alkoxy, arylC1-6 alkoxy, C1 alkyl -6-amino and arylC 1-6 alkylamino, wherein each alkyl, alkoxy or aryl may be optionally substituted with one or more halogen, cyano, C 1-6 alkyl, C 1-6 alkoxy or C 1-6 alkoxy-C 1-6 alkoxy; or R4 and R5 together are X- (CH2) nY, where X and Y are independently selected from the group consisting of CH2, NH and O; n is 1, 2 or 3; and R2 and R3 are defined as described above; A is * NR8-CO, * CO-NR9, * NR8-CS or * CS-NR9, where R8 and R9 are independently selected from the group consisting of hydrogen and C1-6 alkyl, or R8 together with R3 are C2-3 alkylene or CH2CH2O, wherein the oxygen is attached to the phenyl ring, and the * indicates the atom that is attached to the phenyl ring; and R7 is selected from the group that consists of C1-8 alkyl, aryl, heteroaryl, arylC1-6 alkyl, heteroarylC1-6 alkyl, C3-S cycloalkyl, C3-s cycloalkyl C1-6, C1-6 alkoxy, arylC1-6 alkoxy, heteroarylC1-6 alkoxy , C1-6 alkylamino, C1-6 arylalkylamino, C1-6 heteroaryl-alkylamino, di- (C1-6 alkyl) amino, 2,3-dihydrobenzo- [1,4] dioxin-2-yl or adamant-1-yl-methyl, wherein each alkyl and cycloalkyl may be optionally substituted with one or more halogen, cyano, hydroxy, oxo, C1-6 alkoxy or NR10R11, wherein R10 and R11 independently are hydrogen or C1-6 alkyl, or R10 and R11 together with the nitrogen form n an aliphatic ring of 5, 6 or 7 members which may optionally contain another heteroatom selected from N and O, and each aryl may be optionally substituted with one or more halogen, cyano, hydroxy, nitro, C1-6 alkyl, alkoxy C1-6, acyl C1-6, acyloxy C1-6, NR10R11 wherein R10 and R11 independently are hydrogen or C1-6 alkyl, or R10 and R11 together with nitrogen form a 5, 6 or 7 membered aliphatic ring ... |
priorityDate | 2003-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 38.