http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CO-4900049-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_40a92325286ca98dbffa06d2c67ed064 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-40 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-16 |
| filingDate | 1997-09-17-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7ea6ea00d476098bf53ee8de2a9cff0f http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7b6a6b92276cd886e73c21004d2f4c79 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b53acfce28ad60e7afed6ce53e036eca |
| publicationDate | 2000-03-27-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | CO-4900049-A1 |
| titleOfInvention | CERTAIN FUSED PYROLARCARBOXAMIDES; A NEW CLASS OF GABA'S LIGE BRAIN RECEPTORS |
| abstract | A compound of the formula: or pharmaceutically acceptable non-toxic salts thereof wherein: W is aryl or heteroaryl, each of which is optionally substituted with up to 5 groups independently selected from halogen, cyano, hydroxy, alkyl or cycloalkyl with 3 to 7 carbon atoms, amino or mono- or dialkylamino where each alkyl is independently a minor alkyl or a cycloalkyl having 3 to 7 carbon atoms, alkoxy or cycloalkylalkoxy with 3 to 7 carbon atoms, or NR1 COR2, COR2, CONR1 R2 or CO2 R2 where R1 and R2 are the same or different and represent hydrogen or alkyl or cycloalkyl with 3 to 6 carbon atoms; and T is halogen, hydrogen, hydroxyl, amino or alkoxy X is hydrogen, hydroxyl or alkyl; m is 0, 1, or 2; n is 0, 1, or 2; and R3 and R4 are the same or different and are selected from hydrogens, alkyl, COR5 or CO2 R5 where R5 is alkyl or cycloalkyl having 3 to 7 carbon atoms, CONR6 R7, where R6 and R7 are independently selected from hydrogen, alkyl , cycloalkyl having 3 to 7 carbon atoms, phenyl, 2-, 3-, or 4-pyridyl, or NR6 R7 form a heterocyclic group that is morpholinyl, pi-peridinyl, pyrrolidinyl or N-alkylpiperazinyl; or R3-R4 together represent a cyclic part having 3 to 7 carbon atoms. A compound of the formula: where R3 and R4 are the same or different and are selected from hydrogen, alkyl, COR5 or CO2 R5 where R5 is alkyl or cycloalkyl having 3 to 7 carbon atoms, CONR6 R7, where R6 and R7 are independently selected from hydrogen, alkyl, cycloalkyl having 3 to 7 carbon atoms, phenyl, 2-, 3-, or 4-pyridyl, or NR6 R7, form a heterocyclic group that is morpholinyl, piperidinyl, pyrrolidinyl or N- alkylpiperazinyl; or R3 and R4 together represent a cyclic part having 3 to 7 carbon atoms; Y... |
| priorityDate | 1997-09-17-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 25.