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filingDate 2020-10-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2022-08-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-114981266-A
titleOfInvention GABAA positive allosteric modulator compounds, methods for their preparation and uses
abstract Described herein are 2',6-difluoro-5'-[3-(1-hydroxy-1-methylethyl)-imidazo[1,2-b][1,2,4]triazine- 7-yl]biphenyl-2-carbonitrile (TPA023B) or a polymorph of a salt thereof. In one aspect, disclosed herein are crystalline polymorphic salts or co-crystals of TPA023B and phosphoric acid. In another aspect, disclosed herein are crystalline polymorphic salts or co-crystals of TPA023B and sulfuric acid. Also described herein are methods of making and using them.
priorityDate 2019-10-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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