| abstract |
The invention discloses a 4-[α-aryl-β-deuterium-β-(S-ethylformate)]ethylpyridine compound and a preparation method thereof. The technical scheme of the invention is as follows: 4- [α-aryl-β-deuterium-β-(S-ethylformate)]ethylpyridine compounds, which have the following general structural formula: The invention also specifically discloses the specific synthesis process of the 4-[α-aryl-β-deuterium-β-(S-ethylformate)]ethylpyridine compound. The target product obtained by the invention has good regioselectivity, high reaction activity, mild reaction conditions, high deuteration rate of the target product, safety and environmental protection, simple and controllable preparation process, and is suitable for industrial production. |