http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-114685439-A

Outgoing Links

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-06
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-06
filingDate 2020-12-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_38d42de3c60ecb57fe33c3b12110987a
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d0626d5447024660a4c24b09f9392e7f
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c5e715c4c65c5906e8613c3b991efda7
publicationDate 2022-07-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-114685439-A
titleOfInvention A kind of preparation method of lasmiditant
abstract The invention belongs to the technical field of drug synthesis, and in particular relates to a preparation method of lasmidetan. The method for preparing lasmidetan comprises: under the protection of an inert gas, adding a catalyst, a ligand, a base and a solvent A into an airtight In the device, the temperature-controlled reaction is performed, the reaction is completed, the reaction solution is lowered to room temperature, compound SM-1 and compound SM-2 are added, the temperature is raised for reaction, the reaction is completed, and compound I is obtained through post-treatment; the preparation process is simple and convenient, and the obtained compound has high purity , high yield, suitable for industrial production.
priorityDate 2020-12-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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