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publicationDate 2022-01-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-113956272-A
titleOfInvention DNA-PK selective inhibitor and preparation method and application thereof
abstract The application relates to a DNA-PK selective inhibitor shown as a formula (I) and a preparation method and application thereof. The application comprises the application of the compound shown in the formula (I) in preparing a medicament for treating diseases related to DNA-PK. In the preparation process, the compound of the invention is obtained through a series of reactions such as substitution, reduction, cyclization, alkylation and the like. 。
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