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filingDate 2021-07-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-12-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-12-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-113549076-B
titleOfInvention A kind of multi-substituted purine compound and its preparation method and application
abstract The invention discloses a multi-substituted purine compound represented by formula (I) and its pharmaceutically acceptable salt, its preparation method and application. The present invention also discloses that the above-mentioned compound has obvious inhibitory effect on RNA adenosine deaminase 1 (ADAR1), and can be used for preventing and/or treating cancer or tumor-related diseases caused by abnormal activity of this enzyme, especially Prostate cancer, leukemia, breast cancer, multiple myeloma, lung cancer, gastric cancer, ovarian cancer, colon cancer, liver cancer, pancreatic cancer and human glioma and other diseases.
priorityDate 2021-07-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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