http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-113546044-B

Outgoing Links

Predicate Object
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-18
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-44
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-107
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K47-14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K47-44
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-18
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-496
filingDate 2021-07-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-04-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-04-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-113546044-B
titleOfInvention Lurasidone self-microemulsion composition and preparation method thereof
abstract The invention belongs to the technical field of medicines, and particularly discloses a lurasidone self-microemulsion composition and a preparation method thereof, wherein the lurasidone self-microemulsion composition comprises, by weight, 0.1-20 parts of lurasidone, 5-70 parts of an oil phase, 10-70 parts of an emulsifier, and 0-50 parts of a co-emulsifier; the lurasidone self-microemulsion composition forms and releases a microemulsion when contacted with an aqueous medium. The lurasidone free alkali is used as a raw material medicine to prepare the lurasidone self-microemulsion composition, so that the solubility of fat-soluble auxiliary materials is improved, the drug loading rate of a self-microemulsion carrier is improved, and gastrointestinal irritation and other side effects are reduced.
priorityDate 2021-07-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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