abstract |
The present invention discloses a preparation method and application of a novel oxamidox glycoside conjugate bactericide. Amine, N-acetyl-mannosamine and acetylglucosamine are conjugated with oxamidil to obtain a series of oxamidaline glycoside conjugates, the general structural formula of which is shown in I, wherein R is respectively hydroxyl, oxyacetyl, amino , acetamido, R 1 is hydrogen and acetyl. The conjugate of the invention has novel structure, good solubility and antifungal activity, and has the potential to become a new type of green fungicide. |