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filingDate 2019-12-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-04-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-04-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-113024573-B
titleOfInvention Epodophyllotoxin derivative, preparation method and application thereof in preparation of antitumor drugs
abstract The invention discloses an epipodophyllotoxin derivative, which has a structure shown in a general formula I: wherein R is substituted or unsubstituted C4-C15 aryl, substituted or unsubstituted C2-C15 heteroaryl, substituted or unsubstituted C6-C15 fused aryl, and substituted or unsubstituted C4-C-15 fused heteroaryl. Experiments prove that the epipodophyllotoxin derivative disclosed by the invention has good tumor inhibition activity, can be used as an anti-tumor medicament, and is effective on diseases such as leukemia, liver cancer, lung cancer and the like.
priorityDate 2019-12-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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