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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-444
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-12
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-444
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P9-12
filingDate 2019-09-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-08-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-08-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-112384508-B
titleOfInvention Tribicyclic ASK1 inhibitors and their applications
abstract The present invention relates to compounds represented by general formula (I), pharmaceutically acceptable salts, esters or stereoisomers thereof. The present invention also relates to a preparation method of the compound, a pharmaceutical preparation and a pharmaceutical composition comprising the compound. The compounds of the present invention can effectively inhibit the amino acid phosphorylation of ASK1 and inhibit the activation of ASK1; therefore, they can treat and/or prevent diseases mediated by ASK1 and related diseases.
priorityDate 2018-09-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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