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Outgoing Links

Predicate Object
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D231-14
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-655
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D231-14
filingDate 2020-10-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-07-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-07-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-112209878-B
titleOfInvention A kind of cannabinoid receptor light-controlled ligand and its preparation method and application
abstract The invention relates to the field of biotechnology, in particular to a novel cannabinoid receptor light-controlled ligand and a preparation method and application thereof. The cannabinoid receptor light-controlled ligand or its isomer prodrug, solvate, or pharmaceutically acceptable salt, and the structural formula of the cannabinoid receptor light-controlled ligand is: A-linker-B. Among them, A is the transmembrane domain ligand structure, B is the light control element; Linker is a linear subunit that is inactive to the cannabinoid receptor light control ligand. The present invention integrates the cannabinoid receptor ligand with the azobenzene through an appropriate linker, so that the ligand configuration changes under light conditions, thereby regulating the excitation or inhibition state of the cannabinoid receptor.
priorityDate 2020-10-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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