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Outgoing Links

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classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K38-00
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K14-4703
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07K14-47
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K38-17
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00
filingDate 2020-08-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2021-10-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2021-10-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-111944034-B
titleOfInvention Stable polypeptide inhibitor derived from SNAIL1 based on LSD1 substrate and application thereof
abstract The invention provides a polypeptide inhibitor, the amino acid sequence structure of which is shown as follows: the invention also provides application of the polypeptide inhibitor in preparing a medicament for inhibiting the enzymatic activity of LSD 1. The polypeptide can be covalently bound with cysteine (Cys360) near an LSD1 enzyme activity pocket, so that the polypeptide plays a role in inhibiting the activity of LSD1 protease and can be used for in-vivo anti-tumor treatment.
priorityDate 2020-08-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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