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filingDate 2018-09-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a4c63a932af3be45afef94fa546d2dfa
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8ef91377306d2fa3050abcd4f32312de
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publicationDate 2020-10-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-111788208-A
titleOfInvention Tyrantstatin analogs
abstract The present invention provides novel cytotoxic compounds and cytotoxic conjugates comprising these cytotoxic compounds and cell binding agents. More specifically, the present invention relates to novel Tylanstatin A analogs useful as cytotoxic small molecule toxins in antibody-drug conjugates (ADCs). The present invention also relates to compositions comprising these cytotoxic compounds and ADCs, and methods of using these toxins and ADCs to treat pathological conditions, including cancer.
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priorityDate 2017-09-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 761.