http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-111479814-A

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D513-04
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D495-04
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filingDate 2018-12-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e033faa97b6bea099eda1f7b81efa957
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_71366987966af015ef485c197c3a0553
publicationDate 2020-07-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-111479814-A
titleOfInvention Fused pyridines as H-PGDS inhibitors
abstract The application relates to compounds of formula (I), wherein R1, R2, R3, R4, X, Y and A are as defined herein. The compounds of the present invention are inhibitors of hematopoietic prostaglandin D synthase (H-PGDS) and are useful in the treatment of Duchenne muscular dystrophy. Accordingly, the present invention further relates to pharmaceutical compositions comprising the compounds of the present invention. The present invention further relates to methods of inhibiting H-PGDS activity and treating diseases associated therewith using the compounds of the present invention or pharmaceutical compositions comprising the compounds of the present invention.
priorityDate 2017-12-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 519.