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filingDate 2020-03-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-08-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-08-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-111202737-B
titleOfInvention Application of triptolide amide derivatives in the preparation of drugs for the treatment of autoimmune diseases
abstract The invention discloses the use of triptolide amide derivatives represented by formula III or pharmaceutically acceptable salts thereof in preparing medicines for treating autoimmune diseases, wherein R is selected from C1-C6 alkyl groups; Autoimmune diseases are rheumatoid arthritis, systemic lupus erythematosus, and multiple sclerosis. The present invention also discloses a medicine for treating autoimmune diseases, comprising an effective therapeutic dose of triptolide amide derivative or a pharmaceutically acceptable salt thereof and one or more pharmaceutically acceptable excipients. The triptolide amide derivative has high efficiency and low toxicity, can be used as a new type of immunosuppressant with high efficiency and low toxicity, and has the prospect of treating autoimmune diseases, especially rheumatoid arthritis.
priorityDate 2020-03-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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