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classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-5383
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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07H19-24
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07F7-1804
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D413-04
filingDate 2019-08-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2021-04-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2021-04-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-110776501-B
titleOfInvention A kind of preparation method of drug toxin PNU-159682 for antibody drug conjugate and its intermediate
abstract The present invention provides a method for preparing a drug toxin PNU-159682 (morpholinyl anthracycline derivative) for preparing an antibody conjugated drug and an intermediate involved in the preparation method. The preparation method of the present invention improves the stability, practicability and scalability of the process by introducing protective groups and using reagents that are easy to scale up; the preparation method of the present invention reduces the danger and operation difficulty during scaled-up production; preparation The production operation is simple.
priorityDate 2019-08-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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