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http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C327-52
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-04
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00
filingDate 2019-11-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-03-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-03-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-110759891-B
titleOfInvention SET8 lysine methyltransferase inhibitor and intermediate, preparation method and application thereof
abstract The invention provides a SET8 lysine methyltransferase inhibitor and an intermediate, a preparation method and application thereof, wherein the structural general formula of the inhibitor is as follows: the inhibitor has obvious inhibitory activity on SET8 lysine methyltransferase and obvious in-vitro anti-tumor activity, and can be further developed into a targeted anti-tumor medicament with SET8 as a target.
priorityDate 2019-11-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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