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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-04
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D413-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-5377
filingDate 2019-11-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-07-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-07-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-110684022-B
titleOfInvention SET8 lysine methyltransferase inhibitor and its intermediate, preparation method and use
abstract The present invention provides a SET8 lysine methyltransferase inhibitor and its intermediate, preparation method and application. The general structural formula of the inhibitor is as follows, The inhibitor has significant inhibitory activity on SET8 lysine methyltransferase, and also has significant in vitro anti-tumor activity, and can be further developed into a targeted anti-tumor drug targeting SET8.
priorityDate 2019-11-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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