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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00
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filingDate 2019-05-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2021-07-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2021-07-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-110526916-B
titleOfInvention Deuterated Capmatinib compound and application thereof
abstract The invention discloses a deuterated Capmatinib compound and application thereof, and particularly discloses a compound shown as a formula (I) or an optical isomer, a pharmaceutically acceptable salt, a hydrate or a solvate thereof, wherein R is 1 ‑R 16 Each independently selected from H, D, and not all H. The compounds and salts, hydrates or solvates thereof provided by the invention have anticancer activity, better metabolic stability and pharmacokinetic properties and good application prospect.
priorityDate 2018-05-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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