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filingDate 2017-08-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3f12eb4bff22d9cf2b44ffbce26ce06c
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publicationDate 2019-11-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-110494141-A
titleOfInvention Pharmaceutical compositions containing substituted polycyclic pyridone derivatives and prodrugs thereof
abstract The present invention provides pharmaceutical compositions containing the following compounds having antiviral effects. P is a hydrogen atom or a group forming a prodrug; A 1 is CR 1A R 1B , S or O; A 2 is CR 2A R 2B , S or O; A 3 is CR 3A R 3B , S or O; A 4 Each independently is CR 4A R 4B , S or O; wherein, the ring formed by A 1 , A 2 , A 3 , A 4 , a nitrogen atom adjacent to A 1 , and a carbon atom adjacent to A 4 The number of heteroatoms forming ring atoms is 1 or 2; R 1A and R 1B are each independently hydrogen, halogen, or alkyl, etc.; R 2A and R 2B are each independently hydrogen, halogen, or alkyl, etc. R 3A and R 3B are each independently hydrogen, halogen, or alkyl, etc.; R 4A and R 4B are each independently hydrogen, halogen, or alkyl, etc.; R 3A and R 3B optionally together form a non-aromatic carbon Ring or non-aromatic heterocycle; R 1 is a fluorine atom; m is an integer of 1-2, and n is an integer of 1-2.
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Total number of triples: 432.