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filingDate 2018-07-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2023-01-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2023-01-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-110294742-B
titleOfInvention Paracyclic ASK1 inhibitors and applications thereof
abstract The present invention relates to accyclic ASK1 inhibitors and applications thereof, in particular to compounds represented by general formula (I), pharmaceutically acceptable salts, esters or stereoisomers thereof. The present invention also relates to a preparation method of the compound, a pharmaceutical preparation and a pharmaceutical composition containing the compound. The compound of the present invention can effectively inhibit the amino acid phosphorylation of ASK1 and the activation of ASK1; therefore, it can treat and/or prevent ASK1-mediated diseases and related diseases.
priorityDate 2018-03-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415765263
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457280508
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456413165
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID807
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID489547
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456413267
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409901513

Total number of triples: 312.