| abstract |
The invention belongs to the technical field of biological medicines, and particularly relates to a BET protein inhibitor, and a preparation method and application thereof. Compared with the prior art, the invention further improves the structure of the existing BET protein inhibitor to obtain a new-structure BET protein inhibitor, which has better BET protein inhibition activity and good pharmacokinetic property and is expected to be developed into a new-generation high-efficiency low-toxicity BET protein inhibitor. |