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Outgoing Links

Predicate Object
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-517
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-28
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-12
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D239-96
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D405-12
filingDate 2019-03-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-01-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-01-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-109776434-B
titleOfInvention 3-benzyl-6-acylamino-2, 4- (1H,3H) -quinazoline diketone derivative and synthesis method and application thereof
abstract The invention relates to a 3-benzyl-6-acylamino-2, 4- (1H,3H) -quinazoline diketone derivative and a synthesis method and application thereof, belongs to the technical field of medicaments, and relates to a general formula (I), R 1 ,R 2 ,R 3 Are different substituents. The invention discloses the structures and the synthesis methods of the compounds, the inhibitory activity of acetylcholinesterase and the inhibitory activity of phosphodiesterase 5, and the compounds can be further developed into medicaments for treating Alzheimer's disease.
priorityDate 2019-03-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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