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publicationDate 2019-04-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-109562113-A
titleOfInvention Spiro degron for target protein degradation
abstract The present invention provides compounds having spirocyclic E3 ubiquitin ligase targeting moieties (degrons) that can be used as such or linked to targeting ligands for proteins selected for in vivo degradation, the present invention Methods and compositions for their use and methods for their preparation are also provided.
priorityDate 2016-05-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 33.