Predicate |
Object |
assignee |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_ecb7d7f3a37cdebeffcaafcbab7bcb1e |
classificationCPCAdditional |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02A50-30 |
classificationCPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D498-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-554 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-545 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D519-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-438 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-435 |
classificationIPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-527 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D209-54 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D209-96 |
filingDate |
2017-05-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_46fe885aa0fa15c6d61cdc3f96aefd54 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2a40339966abdeaf447b7a6019f97141 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_33de555296bc2c591d895b739ef34437 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_976fe619f7bb3e6a9f263120e87e2b65 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ca103d9b330e58624bb48e9af184ecf0 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e97d69441e27f1656f0639d6a978d7c9 |
publicationDate |
2019-04-02-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber |
CN-109562113-A |
titleOfInvention |
Spiro degron for target protein degradation |
abstract |
The present invention provides compounds having spirocyclic E3 ubiquitin ligase targeting moieties (degrons) that can be used as such or linked to targeting ligands for proteins selected for in vivo degradation, the present invention Methods and compositions for their use and methods for their preparation are also provided. |
priorityDate |
2016-05-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type |
http://data.epo.org/linked-data/def/patent/Publication |