http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-109438318-B
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D209-08 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D209-08 |
| filingDate | 2018-12-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2022-05-03-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2022-05-03-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | CN-109438318-B |
| titleOfInvention | Synthesis method of 3-aryl indole and derivatives thereof |
| abstract | The invention mainly relates to a synthetic method of 3-aryl indole and derivatives thereof, which comprises the following steps: under the action of Lewis acid and S powder, mixing, heating and stirring indole compounds, cyclohexanone compounds and organic solvents for reaction, and then purifying to obtain 3-aryl indole and derivatives thereof. The invention has the following advantages: according to the invention, N-methylindole and cyclohexanone are used as raw materials, and the 3-arylindole and the derivatives thereof are synthesized under the action of Lewis acid and S powder, so that the raw materials are simple, and the synthesis cost is low; the synthetic method provided by the invention does not need transition metal catalysis, and provides a new path for synthesizing the 3-aryl indole compound; the synthesis method has the characteristics of high regioselectivity, simple reaction conditions and the like. |
| priorityDate | 2018-12-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 61.