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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-20
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filingDate 2018-08-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2021-01-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2021-01-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-108938584-B
titleOfInvention Tablet containing VEGF receptor inhibitor Tivozanib salt and preparation method thereof
abstract The invention discloses a tablet containing a VEGF receptor inhibitor Tivozanib salt, which consists of a pharmaceutical active ingredient and an auxiliary material, wherein the pharmaceutical active ingredient is N- { 2-chloro-4- [ (6, 7-dimethoxy-4-quinolyl) oxy ] phenyl } -N' - (5-methyl-3-isoxazolyl) urea (Tivozanib); the auxiliary materials comprise a filling agent, an adhesive, a disintegrating agent and a lubricant, and simultaneously contain lactose and beta-cyclodextrin. The tablet containing the VEGF receptor inhibitor Tivozanib salt is prepared by mixing Tivozanib and beta-cyclodextrin, grinding the mixture to micropowder, adding lactose into the micropowder, continuously grinding the micropowder, adding other auxiliary materials, and tabletting.
priorityDate 2018-08-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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