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publicationDate 2018-11-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-108884058-A
titleOfInvention Macrocyclic Broad Spectrum Antibiotics
abstract Provided herein are antibacterial compounds, wherein in some embodiments the compounds have a broad spectrum of biological activity. In various embodiments, the compounds act by inhibiting an essential protein in bacteria, bacterial type 1 signal peptidase (SpsB). Also provided are pharmaceutical compositions and methods of treatment using the compounds described herein.
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