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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-444
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D405-14
filingDate 2017-11-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2021-11-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2021-11-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-108779100-B
titleOfInvention 3,4-Dipyridylpyrazole derivatives, their preparation method and their application in medicine
abstract The invention relates to 3,4-dipyridylpyrazole derivatives, a preparation method thereof and their application in medicine. Specifically, the present invention relates to a novel 3,4-dipyridylpyrazole derivative represented by the general formula (I), a preparation method thereof, a pharmaceutical composition containing the derivative, and a therapeutic agent thereof, In particular, use as a TGF-β inhibitor and in the preparation of a medicament for the treatment, prevention or reduction of cancer mediated by TGF-β overexpression, wherein each substituent of the general formula (I) is as defined in the description .
priorityDate 2016-11-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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