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classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02P20-55
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C253-20
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C257-14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-13
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C257-14
filingDate 2018-04-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2021-03-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2021-03-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-108727224-B
titleOfInvention Process for preparing intermediates for the synthesis of pharmaceuticals
abstract The invention relates to a preparation method of an intermediate for drug synthesis. Specifically, the present invention relates to a preparation method capable of preparing a compound of the following formula 2 under mild conditions, which is essentially used in the preparation of a compound of the following formula 1, the compound of the following formula 1 being an intermediate for synthesizing a DPP-IV inhibiting therapeutic agent for diabetes, and finally manufacturing the compound of the formula 1 in high yield and purity. Wherein R1, R2, R3, R4, R5 and P1 are defined in the specification.
priorityDate 2017-04-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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