http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-108541255-B

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classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07J1-0011
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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07J43-003
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07J43-00
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filingDate 2016-12-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2019-06-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2019-06-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-108541255-B
titleOfInvention A kind of steroid compound and the composition comprising the compound and application thereof
abstract Composition and its application the present invention provides a kind of steroid compound and comprising the compound.Specifically, steroid compound shown in disclosure of the invention formula (I) and the pharmaceutical composition containing the compound or its crystal form, pharmaceutically acceptable salt, hydrate or solvate, stereoisomer, prodrug, metabolin or isotopic variations.Compound of the present invention can be used as CYP17 enzyme inhibitor, there is better pharmacokinetic parameter characteristic simultaneously, it can be improved the drug concentration of compound in animal body, to improve curative effect of medication and safety, and then it can be used conveniently to prepare the drug for the treatment of Yu CYP17 enzyme related disease (such as prostate cancer).
priorityDate 2016-02-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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