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filingDate 2018-02-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ac0723e9683d76e79ee1d973d439584d
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publicationDate 2018-08-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-108467386-A
titleOfInvention Fused heteroaryl substituted 1,2,4-triazine-3-amine derivatives, preparation method and application in medicine
abstract The invention relates to fused heteroaryl-substituted 1,2,4-triazine-3-amine derivatives, a preparation method thereof and its application in medicine. Specifically, the present invention relates to a fused heteroaryl-substituted 1,2,4-triazine-3-amine derivative represented by general formula (IM), a preparation method thereof and a pharmaceutical composition containing the derivative and its use as a therapeutic agent, especially as an A2a receptor antagonist and in the preparation of a medicament for the treatment of a condition or disorder improved by inhibition of the A2a receptor, wherein the general formula (IM) Each substituent of is the same as defined in the specification.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2019158070-A1
priorityDate 2017-02-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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