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Predicate Object
assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_7f1649e51d42002ff75e3dc3dc8ef653
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-343
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-343
filingDate 2018-06-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_69c8ae7feeb1286822c295aa9eb4d062
publicationDate 2018-08-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-108379250-A
titleOfInvention Chloranthalactone A is used as the biomedical uses of 1 inhibitor of indoleamine 2,3-dioxygenase
abstract The invention discloses chloranthalactone A to be used as indoleamine 2, the biomedical uses of 3 dioxygenase, 1 inhibitor.It is a discovery of the invention that chloranthalactone A, chloranthalactone C, chloranthalactone D, chloranthalactone E and chloranthalactone F are indoleamine 2, effective inhibitor of 3 dioxygenases 1 (IDO1).Numerous studies show that the unconventionality expression of IDO1 is related with tumour cell escape immune system, therefore IDO1 is inhibited to be expected to become a kind of novel tumor therapeutic strategy.Currently, indoximod, epacadostat and NLG919 are the IDO1 inhibitor in clinical investigation phase, in addition there are multiple inhibitor to be in the biological activity test stage.IDO1 inhibitor has a extensive future.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-111035623-B
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-111035623-A
priorityDate 2018-06-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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