Predicate |
Object |
classificationCPCAdditional |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02A50-30 |
classificationCPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P33-06 |
classificationIPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D417-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P33-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-513 |
filingDate |
2016-11-24-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
grantDate |
2021-08-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationDate |
2021-08-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber |
CN-108290860-B |
titleOfInvention |
Iminotetrahydropyrimidinone derivatives as PLASMEPSIN V inhibitors |
abstract |
A series of 2-imino-6-methyltetrahydropyrimidin-4 (1H) -one derivatives, substituted in the 6-position by a phenyl group which in turn is meta-substituted by an optionally substituted unsaturated fused bicyclic ring system containing at least one nitrogen atom, are useful as selective inhibitors of plasmepsin V activity as medicaments, in particular in the treatment of malaria. |
priorityDate |
2015-11-25-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type |
http://data.epo.org/linked-data/def/patent/Publication |