http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-107922381-B

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-18
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-444
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-00
filingDate 2016-10-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2020-10-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2020-10-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-107922381-B
titleOfInvention Pyridine or pyrimidine derivatives
abstract The invention relates to compounds of formula (I), wherein R 1’ Is methyl; r 1 Is methyl, ethyl, CF 3 、CH 2 OH, cyclopropyl or cyano, or R 1’ And R 1 May together form a1, 1-dioxo-tetrahydro-thiophen-3-yl ring; r 2 Is hydrogen, methyl, ethyl, isopropyl, tert-butyl, cyclopropyl, cyclopropylmethyl or hydroxymethyl; r 3 Is Cl, F, CF 3 Methyl, methoxy or cyclopropyl; r 4 Is hydrogen, methyl, F or Cl; x is N or CH; y is N or CH; provided that X and Y are not both CH; or to a pharmaceutically acceptable salt or acid addition salt, to a racemic mixture, or to its corresponding enantiomer and/or optical isomer and/or stereoisomer thereof. The compounds of formula (I) may be used for the treatment of psychotic disorders such as schizophrenia, bipolar disorder, obsessive-compulsive disorder or autism spectrum disorder.
priorityDate 2015-10-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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