http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-107674016-B

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filingDate 2016-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2020-06-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2020-06-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-107674016-B
titleOfInvention Preparation method of telaprevir intermediate and intermediate thereof
abstract The invention discloses a preparation method of a telaprevir intermediate and an intermediate thereof. The invention specifically discloses a preparation method of a compound shown as a formula 6, which comprises the following steps of carrying out the following reaction on a compound shown as a formula 7 or a formula 5 under the action of an aqueous solution of acid and at the temperature of 50-100 ℃; the method has the advantages of simple operation, lower cost, higher yield, better purity and easy realization of industrial production.
priorityDate 2016-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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