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publicationDate 2018-01-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-107531668-A
titleOfInvention Therapeutic pyridazine compounds and uses thereof
abstract The present invention relates to compounds of formula (I) and salts thereof, as well as compositions and uses thereof, wherein: R 1 -R 4 has any value defined in the specification. The compounds are useful as inhibitors of BRG1, BRM and/or PB1. The present invention also includes a pharmaceutical composition comprising a compound of formula (I) or a pharmaceutically acceptable salt thereof, and a method for using the above-mentioned compound and salt to treat various BRG1-mediated disorders, BRM-mediated disorders and/or PB1-mediated disorders method.
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