http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-107513093-A

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07J41-0066
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07J41-00
filingDate 2017-09-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_86b9b941cdef257e509c17ab579e7203
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c2a30d3da1cdf8c47a4a153d8dfaf11d
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publicationDate 2017-12-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-107513093-A
titleOfInvention The preparation method of epristeride intermediate and preparation method thereof, epristeride
abstract The present invention relates to drug field, in particular to the preparation method of a kind of epristeride intermediate and preparation method thereof, epristeride.A kind of preparation method of epristeride intermediate, it comprises the following steps:Compound 3 and alkaline reagent sulfonating reaction generation compound 4;Compound 3 and alkaline reagent sulfonating reaction generation compound 4, reaction conversion is single, avoids column chromatography for separation;The alkaline reagent that course of reaction uses is readily available, and reaction condition is gentle.And reduce unit operation, the production cycle is shortened, improves production efficiency.Production efficiency is high, improves economic benefit.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-111624291-A
priorityDate 2017-09-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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