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filingDate 2016-02-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2021-06-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2021-06-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-107428752-B
titleOfInvention Homemade chemokine-inhibiting compounds
abstract The present invention relates to compounds of formula I , wherein A1, A2, A3, R1, R2, R3 , R4, R5 , R6 , L , Ar and Q are each as defined herein. The compounds of the present invention are inhibitors of autotaxin (ATX) enzymatic activity. The present invention also relates to processes for preparing these compounds, pharmaceutical compositions containing them, and their use in the treatment of proliferative disorders such as cancer, and other diseases or conditions in which ATX activity is implicated (eg, fibrosis).
priorityDate 2015-02-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122485170
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8ZV53
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO77762
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2SSX9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415996935
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122485171
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID177913
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414239701
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2733084
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9CHX5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID425994407
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122485172
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF1N1G1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8VVL0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3KYH2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID140819
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4L800
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13157
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5QWC7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP47280
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122445541
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ31ZS8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID510618
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66774
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24577
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122445542
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281572
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122199235
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2RZH4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122445528
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122485162
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7Z9S5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421016707
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP37997
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID412156787
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122445529
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ64702
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403441
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2TA25
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122445530
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122445531
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID481131
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ20845
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122485150
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB8E001
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411272810
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID134170299
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09476
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5PXD0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122445519
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ08867
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122485153
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID134170300
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09477
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419540924
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122485154
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8P126
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422000484
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ57NR0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP34331
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408091139
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122485155
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122445521
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8018
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9N2L7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413929623
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID159324
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457814460
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122445523
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9910224
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411473989
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420303774
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP60569
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB3PM40
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23331
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67965
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5PCT4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122445525
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23335
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP52304
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67968
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID75555
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135400182
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1024199
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122445526
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8NVG5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67969
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457797616
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12978
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57363
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP46649
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419486648
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122485075
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67970
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81423
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP62205
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393353
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67971
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID380430
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP46652
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID32876
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122445577
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6484228
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67973

Total number of triples: 1364.