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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-16
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-34
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P3-10
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-16
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K47-34
filingDate 2016-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2020-11-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2020-11-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-107405307-B
titleOfInvention Exenatide microsphere preparation and preparation method thereof
abstract The invention discloses an exenatide microsphere preparation, which comprises the following components in percentage by weight: 3% -10% of exenatide or exenatide salt and 88% -97% of PLGA, wherein the PLGA is a mixture of low-viscosity PLGA and high-viscosity PLGA, and the weight ratio of the low-viscosity PLGA to the high-viscosity PLGA is 1: 1-9: 1. the invention also provides an O/W preparation method of the preparation. The exenatide microsphere preparation prepared by the invention has the advantages of small burst release, short release lag phase and C max /C ave Low, is beneficial to reducing the risk caused by the large fluctuation of the blood concentration when the type II diabetes is treated, and has better clinical application prospect.
priorityDate 2015-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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