http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-107151242-B
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-653 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-50 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4178 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4196 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D409-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01P3-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-50 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P31-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-653 |
| filingDate | 2016-03-02-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2020-05-22-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2020-05-22-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | CN-107151242-B |
| titleOfInvention | 2-azolothiochromone compound, synthesis method thereof and application thereof in preparation of antifungal drugs |
| abstract | The invention relates to a 2-azolothiazolone compound (formula I) with the following structure, wherein R 1 Is substituted by hydrogen or C 1 ‑C 3 An alkyl-substituted five-membered azodicarbonyl ring; r 2 Is hydroxy, C 1 ‑C 6 Hydrocarbyloxy group of (C) 1 ‑C 6 With hydrocarbon amino group, C 1 ‑C 6 A hydrocarbon group of (C), a phenyl group 1 ‑C 6 Hydrocarbyloxy-substituted phenyl, phenoxy, by 1 or more C 1 ‑C 6 Alkoxy-substituted phenoxy; r 3 、R 4 、R 6 Each independently selected from hydrogen, fluorine, chlorine, bromine or iodine; r 5 Selected from hydrogen, fluorine, chlorine, bromine, iodine, C 1 ‑C 6 Hydrocarbyloxy group of (C) 1 ‑C 6 With 1 or more C, a phenoxy group 1 ‑C 6 A phenoxy group substituted with a hydrocarbon group or a hydrocarbonoxy group. The compound of the invention has the application of preparing antifungal medicines, and has stronger bacteriostatic activity on common pathogenic fungi and deep fungal infectionLow toxicity, high stability and broad antifungal spectrum. |
| priorityDate | 2016-03-02-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 119.