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filingDate 2015-11-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2019-06-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2019-06-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-107001374-B
titleOfInvention 1-[2-(Aminomethyl)benzyl]-2-thio-1,2,3,5-tetrahydro-4H-pyrrolo[3,2-D] as a myeloperoxidase inhibitor Pyrimidine-4-one
abstract Disclosed herein are certain 1-[2-(aminomethyl)benzyl]-2-thio-1,2,3,5-tetrahydro-4H-pyrrolo[3,2- d] a pyrimidin-4-one compound, and pharmaceutically acceptable salts thereof, as well as compositions containing these compounds and the use of these compounds and compositions in therapy. These compounds are inhibitors of the enzyme MPO and are therefore particularly useful in the treatment or prevention of cardiovascular disorders, such as heart failure and coronary artery disease related disorders.
priorityDate 2014-12-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 530.