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filingDate 2015-09-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2019-08-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2019-08-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-106795139-B
titleOfInvention Aminopyridyloxypyrazole compounds
abstract The present invention relates to novel aminopyridyloxypyrazole compounds that inhibit the activity of transforming growth factor beta receptor 1 (TGFβR1), pharmaceutical compositions comprising said compounds and use of said compounds for the treatment of cancer, preferably colon cancer, black A method for melanoma, hepatocellular carcinoma, renal carcinoma, glioblastoma, pancreatic cancer, myelodysplastic syndrome, lung and gastric cancer and/or fibrosis, preferably liver fibrosis and chronic kidney disease.
priorityDate 2014-10-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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