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classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02P20-55
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C51-08
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C59-48
filingDate 2016-11-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2017-12-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2017-12-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-106565467-B
titleOfInvention A kind of preparation method of antiallergic bilastine intermediate
abstract The invention discloses a kind of preparation method of antiallergy new drug bilastine intermediate, more difficult quaternary carbon atom is built using gentle addition reaction, carboxylic group is introduced at room temperature with very cheap and easily-available raw material, purify the research of progress to it using distinctive two phasic property of carboxylic acid simultaneously, so that the expensive metallic catalyst avoided in building-up process, it it also avoid the implementation condition of harshness, it is gentle so as to provide a reaction condition, it is easy to operate, synthesis cost is cheap, is adapted to the preparation method of the Bilastine intermediates of large-scale production.
priorityDate 2016-11-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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