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classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02A50-30
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D285-36
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P31-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D285-36
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-554
filingDate 2016-10-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-09-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2018-09-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-106543102-B
titleOfInvention 1,5- benzothiazepines analog derivative and its application
abstract The invention discloses application of the 1,5 benzothiazepines analog derivatives in antibacterials with general formula I: In Formulas I, R 1 ,R 2 ,R 3, R 4 ,R 5 ,R 6 ,R 7 ,R 8 ,R 9 It is each independently OCH 3 , OH, H, CF 3 , halogen;Y is respectively F, Br, Cl, CF 3 ,CHF 2 ,CH 2 F,CF 2 Cl,CF 3 CF 2 ,CHF 2 CF 2 .The compound of the present invention has apparent inhibiting effect, can be used for preparing antibacterials to Candida albicans, Methicillin-resistant Staphylococcus color staphylococcus, Escherichia coli and Pseudomonas aeruginosa.
priorityDate 2016-10-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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