http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-105646469-B
Outgoing Links
Predicate | Object |
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classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D413-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P31-04 |
filingDate | 2014-11-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
grantDate | 2019-06-04-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationDate | 2019-06-04-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | CN-105646469-B |
titleOfInvention | A kind of oxazolidinones antimicrobial phosphate and preparation method thereof |
abstract | The invention discloses a kind of oxazolidinones antimicrobial phosphate and preparation method thereof, be related to oxazolidinones antimicrobial ( S )‑ N [[3- [the fluoro- 4- of 3- (4- (2- pyridine) -1 H Pyrazol-1-yl) phenyl] -2- oxo -5- oxazolidinyl] methyl]-acetamide diphosphate preparation and characterization.Problem to be solved by this invention be improve ( S )‑ N [[3- [the fluoro- 4- of 3- (4- (2- pyridine) -1 H Pyrazol-1-yl) phenyl] -2- oxo -5- oxazolidinyl] methyl] dissolubility of-acetamide in water, by preparing its stable diphosphate, according to the present invention ( S )‑ N [[3- [the fluoro- 4- of 3- (4- (2- pyridine) -1 H Pyrazol-1-yl) phenyl] -2- oxo -5- oxazolidinyl] methyl]-acetamide diphosphate have excellent water solubility, the antibacterial activity of drug in vivo can be effectively improved. |
priorityDate | 2014-11-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 55.