http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-105377834-B

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filingDate 2014-04-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-04-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2018-04-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-105377834-B
titleOfInvention Derivatives of dolastatin 10 and auristatin
abstract The present invention relates to compounds of the following formula (I) wherein: -R 1 is H or OH, -R 2 is (C 1 -C 6 ) alkyl, COOH, COO-((C 1 -C 6 ) alkyl) or thiazole group, -R 3 is H or (C 1 -C 6 ) alkyl, and -R 4 is aryl -(C 1 -C 6 ) substituted by one or more groups selected from OH and NR 9 R 10 groups C 8 ) alkyl, or a pharmaceutically acceptable salt, hydrate or solvate thereof, and uses thereof, especially for treating cancer, a pharmaceutical composition containing the same, and a preparation method thereof.
priorityDate 2013-04-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 73.