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filingDate 2014-03-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2019-04-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2019-04-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-105324117-B
titleOfInvention Polysubstituted aromatic compounds as serine protease inhibitors
abstract In particular, the present invention provides polysubstituted aromatic compounds comprising substituted pyrazolyl or substituted triazolyl, useful for inhibiting kallikrein. Also provided are pharmaceutical compositions. Also provided are methods for the treatment and prevention of certain diseases or conditions amenable to treatment or prevention by inhibition of kallikrein.
priorityDate 2013-03-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135565674
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1127
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID37662
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO61608
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424526205
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419548914
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419545923
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456087266
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419590872
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID43736
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP36373
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8WUW1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID441478
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419485447
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO61309
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25048
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419552660
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID407998
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ03352
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP36376
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID931
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454339991
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID744785
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID313
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP08611
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP32261
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP36369
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID32876
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP32262
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54678486
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ91VR8
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2KJ63
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10553
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419532030
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457637874
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11587
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457637794
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2091
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID7422
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID90338
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420129773
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID408211
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5270
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID407126721
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394295
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448766806
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8005
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO01945
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP83906
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ29485
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ43880
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID290757
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135552039
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421463122
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2146
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394314
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13726
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID83785
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID136071
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP84122
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID7116
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID62493
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419511492
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID152951
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID288001
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457193112
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID462
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24594
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281572
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420166891
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GKR0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10476

Total number of triples: 393.