http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-104903327-B

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-5025
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P29-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04
filingDate 2014-01-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2016-09-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2016-09-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-104903327-B
titleOfInvention For treating the pyrido-as autotaxin inhibitor or the pyrrolo--fused pyrimidine derivative of pain
abstract The present invention provides the compound of Formulas I, its officinal salt: Wherein X is key or CH 2 ;R is selected from With ;R 1 And R 2 It is each independently selected from CH and N;R 3 It is H or CH 3 ;R 4 It is H or CH 3 ;L is selected from O (CH 2 ) 3 ‑、‑C(O)NH(CH 2 ) 2 ‑、‑CH 2 C(O)NH(CH 2 ) 2 ‑、‑(CH 2 ) 3 N(C(O)CH 3 )CH 2 ‑、‑(CH 2 ) 2 N(C(O)CH 3 )CH 2 ‑、‑(CH 2 ) 3 NH‑、(CH 2 ) 2 OCH 2 ‑、‑(CH 2 ) 4 ‑、‑(CH 2 ) 2 NHCH 2 ‑、‑(CH 2 ) 3 O and CH 2 O(CH 2 ) 2 ‑.The compound of the present invention is autotaxin inhibitor.
priorityDate 2013-01-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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